SCHEMBL4352985

SCHEMBL4352985

O=C(Nc1ccc(Oc2ccccc2)cc1)Nc1ccc(O)c(F)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.58
CA1 P00915 4/20 0.58
CA2 P00918 4/20 0.58
CA9 Q16790 4/20 0.58
PNLIP P16233 2/20 0.54
FAAH O00519 1/20 0.53
HPGD P15428 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
PGR P06401 1/20 0.51
MAPT P10636 3/20 0.50
MEN1 O00255 2/20 0.50
LMNA P02545 2/20 0.50
KMT2A Q03164 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
RAF1 P04049 2/20 0.49
MAPK13 O15264 1/20 0.49
MAPK12 P53778 1/20 0.49
MAPK11 Q15759 1/20 0.49
MAPK14 Q16539 1/20 0.49
EPHX1 P07099 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6229951 0.99 CA12 (0.60) CA12CA1CA2CA9PNLIP
SCHEMBL4351601 0.88 MAOA (0.59) SMN1; SMN2MAPTMEN1LMNAKMT2A
SCHEMBL4346263 0.87 CA12 (0.56) CA12CA1CA2CA9PNLIP
SCHEMBL6673220 0.86 CA12 (0.55) CA12CA1CA2CA9PNLIP
SCHEMBL4354589 0.83 MEN1 (0.61) CA12CA1CA2CA9PNLIP
SCHEMBL30053559 0.83 CA12 (0.73) CA12CA1CA2CA9PNLIP
SCHEMBL6252145 0.82 CA12 (0.60) CA12CA1CA2CA9PNLIP
SCHEMBL21295380 0.81 CA12 (0.71) CA12CA1CA2CA9PNLIP
SCHEMBL6229953 0.80 FAAH (0.48) CA12CA1CA2CA9PNLIP
SCHEMBL4347138 0.80 EPHX2 (0.71) FAAHHPGDMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed