SCHEMBL434748

SCHEMBL434748

Fc1cc(Cl)ccc1-c1cc[c]c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 3/20 0.36
KMO O15229 2/20 0.35
EGLN2 Q96KS0 1/20 0.34
CNR1 P21554 1/20 0.34
FASN P49327 1/20 0.34
CLK1 P49759 1/20 0.33
ESR1 P03372 2/20 0.33
ESR2 Q92731 2/20 0.33
AHR P35869 1/20 0.32
BCHE P06276 1/20 0.32
HSD11B1 P28845 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
APP P05067 1/20 0.32
S100A4 P26447 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL432713 0.86 TTR (0.44) GRM2CNR1ESR1ESR2APP
SCHEMBL433433 0.86 GRM2 (0.36) GRM2KMOEGLN2CNR1FASN
SCHEMBL15637653 0.81 ESR1 (0.34) ESR1ESR2
SCHEMBL432623 0.81 AHR (0.52) AHRHSD11B1
SCHEMBL432735 0.80 PTPRC (0.43) HSD11B1
SCHEMBL434681 0.79 GRM2 (0.41) GRM2KMOEGLN2CNR1FASN
SCHEMBL17514851 0.79 AHR (0.39) GRM2KMOEGLN2CNR1FASN
SCHEMBL17514488 0.79 CTSD (0.36) GRM2KMOEGLN2CNR1FASN
SCHEMBL2052439 0.79 GRM5 (0.33) CNR1
SCHEMBL15637040 0.78 TP53 (0.38) AHRS100A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016026830-A1 NOVEL FUNGICIDAL PYRAZOLE DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-02-25 WO disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed