SCHEMBL434931

SCHEMBL434931

O=C(Nc1ccc(C(F)(F)F)nc1OC1CN(CC=Cc2ccc(Cl)cc2)C1)c1ccnc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
P2RX7 Q99572 1/20 0.34
MCHR1 Q99705 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33
SCN9A Q15858 1/20 0.33
PROKR1 Q8TCW9 1/20 0.33
S1PR3 Q99500 1/20 0.32
EBP Q15125 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
RAF1 P04049 1/20 0.32
SMARCA2 P51531 1/20 0.32
SMARCA4 P51532 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL432023 1.00 GRM5 (0.34) GRM5MEN1KMT2AP2RX7MCHR1
SCHEMBL432153 0.88 GSK3B (0.35) MCHR1SCN9APROKR1EBPSIGMAR1
SCHEMBL432154 0.88 GSK3B (0.35) MCHR1SCN9APROKR1EBPSIGMAR1
SCHEMBL431257 0.87 MCHR1 (0.34) MEN1KMT2AMCHR1SCN9APROKR1
SCHEMBL431256 0.87 MCHR1 (0.34) MEN1KMT2AMCHR1SCN9APROKR1
SCHEMBL460699 0.87 GRM5 (0.34) GRM5MEN1KMT2AP2RX7CYP1A2
SCHEMBL460698 0.87 GRM5 (0.34) GRM5MEN1KMT2AP2RX7CYP1A2
SCHEMBL433488 0.86 EBP (0.36) MEN1KMT2AMCHR1SCN9APROKR1
SCHEMBL432987 0.86 MAPT (0.37) MCHR1SCN9APROKR1EBPSIGMAR1
SCHEMBL432986 0.86 MAPT (0.37) MCHR1SCN9APROKR1EBPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012366-A1 PESTICIDAL 3-(ARYLOXY)AZACYCLOALKANES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-01-26 WO claimed
WO-2012012366-A1 PESTICIDAL 3-(ARYLOXY)AZACYCLOALKANES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-01-26 WO disclosed