SCHEMBL4350019

SCHEMBL4350019

Oc1ccc(NC(=S)NC2CCCCC2)cc1Cl

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 11/20 0.79
MEN1 O00255 7/20 0.79
KMT2A Q03164 7/20 0.79
MAPT P10636 7/20 0.79
LMNA P02545 6/20 0.79
NPSR1 Q6W5P4 3/20 0.79
HTT P42858 3/20 0.79
ALOX12 P18054 2/20 0.79
CYP1A2 P05177 3/20 0.64
CYP2C19 P33261 3/20 0.64
CYP3A4 P08684 2/20 0.64
CYP2D6 P10635 1/20 0.64
RAB9A P51151 6/20 0.59
GAA P10253 3/20 0.59
NPC1 O15118 5/20 0.58
MAPK1 P28482 2/20 0.57
ALDH1A1 P00352 3/20 0.56
HPGD P15428 1/20 0.56
BLM P54132 1/20 0.56
POLB P06746 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11845603 0.88 SMN1; SMN2 (1.00) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL4348625 0.84 SMN1; SMN2 (0.71) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL4347357 0.83 SMN1; SMN2 (0.62) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL4359761 0.83 RAB9A (0.73) SMN1; SMN2MEN1KMT2ALMNAHTT
SCHEMBL6565598 0.82 SMN1; SMN2 (0.68) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL28756963 0.81 SMN1; SMN2 (0.83) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL11697622 0.80 NPSR1 (1.00) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL4348605 0.80 SMN1; SMN2 (0.55) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL12239184 0.79 S1PR1 (0.57) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL26123831 0.78 MEN1 (1.00) SMN1; SMN2MEN1KMT2AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed