SCHEMBL4350040

SCHEMBL4350040

COc1ccc(Sc2ccccc2CNc2cc(Cl)c(O)c(Cl)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.58
MEN1 O00255 4/20 0.58
POLB P06746 3/20 0.58
MMP2 P08253 5/20 0.51
MMP9 P14780 5/20 0.51
MMP12 P39900 5/20 0.51
MMP14 P50281 1/20 0.51
MAPT P10636 4/20 0.43
KDM4E B2RXH2 3/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
ALOX15 P16050 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
MAOB P27338 1/20 0.40
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6226094 0.91 KMT2A (0.51) KMT2AMEN1POLBMMP2MMP9
SCHEMBL4347108 0.90 KMT2A (0.50) KMT2AMEN1POLBMMP2MMP9
SCHEMBL4349041 0.90 MEN1 (0.50) KMT2AMEN1POLBMMP2MMP9
SCHEMBL4350028 0.89 MEN1 (0.56) KMT2AMEN1POLBMMP2MMP9
SCHEMBL4349243 0.87 MAPT (0.46) KMT2AMEN1POLBMAPTKDM4E
SCHEMBL4349840 0.87 SLC6A4 (0.48) KMT2AMEN1POLBMAPTKDM4E
SCHEMBL4351063 0.86 SMN1; SMN2 (0.43) KMT2AMEN1POLBMAPTKDM4E
SCHEMBL4359446 0.86 MEN1 (0.58) KMT2AMEN1POLBMMP2MMP9
SCHEMBL4353810 0.86 MEN1 (0.58) KMT2AMEN1POLBMMP2MMP9
SCHEMBL4345485 0.85 KMT2A (0.55) KMT2AMEN1POLBMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed