SCHEMBL4349243

SCHEMBL4349243

Cc1ccc(Sc2ccccc2CNc2cc(Cl)c(O)c(Cl)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.46
SLC6A4 P31645 5/20 0.40
SLC6A3 Q01959 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
SLC6A2 P23975 3/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
CYP2D6 P10635 2/20 0.39
GFER P55789 1/20 0.39
CYP3A4 P08684 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALOX15 P16050 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PLA2G1B P04054 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6225098 0.90 MAPT (0.40) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4349840 0.90 SLC6A4 (0.48) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4351063 0.90 SMN1; SMN2 (0.43) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4351627 0.89 MAPT (0.39) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4345579 0.89 MAPT (0.39) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4345804 0.88 MAPT (0.50) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4350040 0.87 KMT2A (0.58) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4345899 0.86 MEN1 (0.47) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4350338 0.85 MAPT (0.46) MAPTSLC6A4SLC6A3MEN1KMT2A
SCHEMBL4350004 0.85 MAPT (0.46) MAPTSLC6A4SLC6A3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed