SCHEMBL4350367

SCHEMBL4350367

CC(C)(C)NC(=O)Nc1cc(Cl)c(O)c(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.62
NPC1 O15118 3/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
RAB9A P51151 2/20 0.50
POLB P06746 3/20 0.49
MAPK1 P28482 1/20 0.49
KDM4E B2RXH2 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
DHODH Q02127 1/20 0.46
TP53 P04637 1/20 0.46
GAA P10253 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
HSD17B10 Q99714 1/20 0.46
APEX1 P27695 1/20 0.44
EPHX1 P07099 1/20 0.43
EPHX2 P34913 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12846674 0.89 HTT (0.55) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL4359277 0.85 HTT (0.51) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL6567241 0.82 EPHX1 (0.59) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL4341979 0.82 POLB (0.54) HTTNPC1MEN1KMT2APOLB
SCHEMBL21116152 0.81 HTT (0.61) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL4342347 0.81 HTT (0.70) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL6526431 0.81 HTT (0.47) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL17849580 0.81 MEN1 (0.60) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL4351163 0.79 HTT (0.58) HTTNPC1MEN1KMT2ARAB9A
SCHEMBL4343700 0.79 HTT (0.50) HTTMEN1KMT2APOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed