SCHEMBL4351774

SCHEMBL4351774

Oc1c(Cl)cc(NCc2cccc(C(F)(F)F)c2)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.54
FFAR4 Q5NUL3 1/20 0.54
LMNA P02545 2/20 0.50
GAA P10253 2/20 0.50
P2RX7 Q99572 1/20 0.50
MEN1 O00255 1/20 0.50
PLA2G1B P04054 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ATG4B Q9Y4P1 1/20 0.50
HPGD P15428 1/20 0.50
RXFP1 Q9HBX9 1/20 0.48
KCNN3 Q9UGI6 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355530 0.86 FFAR1 (0.55) FFAR1FFAR4LMNAGAAP2RX7
SCHEMBL4352193 0.84 FFAR1 (0.55) FFAR1FFAR4GAAMEN1PLA2G1B
SCHEMBL4348617 0.82 MEN1 (0.53) FFAR1FFAR4LMNAGAAP2RX7
SCHEMBL4345824 0.82 RXFP1 (0.53) FFAR1FFAR4LMNAGAAP2RX7
SCHEMBL5226860 0.81 FFAR1 (0.61) FFAR1FFAR4LMNAGAAP2RX7
SCHEMBL631859 0.79 MEN1 (0.55) FFAR1FFAR4LMNAGAAP2RX7
SCHEMBL4242744 0.79 FFAR1 (0.66) FFAR1FFAR4LMNAGAAMEN1
SCHEMBL4347062 0.78 P2RX7 (0.48) P2RX7MEN1CYP1A2CYP3A4CYP2D6
SCHEMBL4349831 0.77 RXFP1 (0.46) FFAR1FFAR4LMNAGAAP2RX7
SCHEMBL4341276 0.76 FFAR1 (0.56) FFAR1FFAR4GAAMEN1PLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed