SCHEMBL4351892

SCHEMBL4351892

Oc1c(Cl)cc(NC(=S)Nc2ccccc2)cc1Cl

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.63
CYP3A4 P08684 1/20 0.63
TAS2R38 P59533 1/20 0.63
HSD17B10 Q99714 1/20 0.63
RAB9A P51151 3/20 0.58
NPC1 O15118 2/20 0.58
HTT P42858 1/20 0.58
KMT2A Q03164 5/20 0.58
MAOB P27338 3/20 0.58
GAA P10253 2/20 0.58
MAOA P21397 2/20 0.58
LMNA P02545 1/20 0.58
MEN1 O00255 3/20 0.53
NOX1 Q9Y5S8 2/20 0.53
MAPT P10636 3/20 0.52
KDM4E B2RXH2 1/20 0.51
MAPK1 P28482 1/20 0.50
ALOX12 P18054 1/20 0.49
PPARG P37231 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347956 0.85 ALDH1A1 (0.58) ALDH1A1RAB9ANPC1HTTKMT2A
SCHEMBL4354098 0.83 ALDH1A1 (0.47) ALDH1A1CYP3A4TAS2R38HSD17B10RAB9A
SCHEMBL4343605 0.82 KMT2A (0.59) ALDH1A1CYP3A4TAS2R38HSD17B10RAB9A
SCHEMBL4346849 0.82 ALDH1A1 (0.68) ALDH1A1CYP3A4TAS2R38HSD17B10RAB9A
SCHEMBL5450586 0.81 ALDH1A1 (0.71) ALDH1A1CYP3A4TAS2R38HSD17B10RAB9A
SCHEMBL4342381 0.81 KMT2A (0.68) RAB9ANPC1HTTKMT2AMAOB
SCHEMBL4342470 0.81 IDO1 (0.60) ALDH1A1CYP3A4HSD17B10HTTKMT2A
SCHEMBL4355796 0.80 MAPT (0.66) ALDH1A1RAB9ANPC1HTTKMT2A
SCHEMBL6815028 0.80 GAA (0.60) ALDH1A1CYP3A4HTTKMT2AMAOB
SCHEMBL132620 0.79 ALDH1A1 (1.00) ALDH1A1CYP3A4TAS2R38HSD17B10RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed