SCHEMBL435210

SCHEMBL435210

Fc1[c]cccc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.41
AHR P35869 1/20 0.40
CRHR1 P34998 4/20 0.39
HSP90AA1 P07900 2/20 0.37
HSP90AB1 P08238 2/20 0.37
TP53 P04637 3/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
KDM4E B2RXH2 2/20 0.36
S100A4 P26447 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
SRD5A2 P31213 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
DPP4 P27487 1/20 0.35
GPR3 P46089 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433432 0.86 GRM2 (0.38) HSD11B1S100A4GPR3
SCHEMBL17514776 0.86 HSD11B1 (0.43) HSD11B1TP53NPC1RAB9AGPR3
SCHEMBL432622 0.81 AHR (0.42) HSD11B1AHRCRHR1TP53NPC1
SCHEMBL5182077 0.81 PDK2 (0.36) HSD11B1AHRALDH1A1
SCHEMBL3790757 0.81 CYP2A6 (0.41) HSD11B1HSP90AA1HSP90AB1TP53NPC1
SCHEMBL15636309 0.79 AHR (0.40) HSD11B1AHRCRHR1HSP90AA1HSP90AB1
SCHEMBL15637459 0.78 HSD11B1 (0.42) HSD11B1AHRCRHR1TP53NPC1
SCHEMBL436977 0.77 HSD11B1 (0.43) HSD11B1AHRHSP90AA1HSP90AB1TP53
SCHEMBL13728896 0.76 RECQL (0.41) SMN1; SMN2KDM4EALDH1A1HPGDNPSR1
SCHEMBL433163 0.76 CYP1A2 (0.38) AHRTP53NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
EP-0133805-A2 Triazole antifungal agents Pfizer Limited (GB) 1985-03-06 EP disclosed