Tofisopam

Tofisopam

SCHEMBL43522

CCC1C(C)=NN=C(c2ccc(OC)c(OC)c2)c2cc(OC)c(OC)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 1.00
PDE4A P27815 2/20 1.00
MEN1 O00255 1/20 1.00
CHRM1 P11229 1/20 1.00
PDE4D Q08499 1/20 1.00
PDE3A Q14432 1/20 1.00
CA2 P00918 1/20 0.38
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 5/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HSD17B10 Q99714 2/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.36
ATM Q13315 1/20 0.36
MAPT P10636 2/20 0.36
HTT P42858 2/20 0.36
ALOX5 P09917 1/20 0.35
EPHX2 P34913 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
BRD4 O60885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Levotofisopam SCHEMBL5431173 1.00 KMT2A (1.00) KMT2APDE4AMEN1CHRM1PDE4D
Dextofisopam SCHEMBL236796 1.00 KMT2A (1.00) KMT2APDE4AMEN1CHRM1PDE4D
Tofisopam SCHEMBL29832594 1.00 KMT2A (1.00) KMT2APDE4AMEN1CHRM1PDE4D
Dextofisopam SCHEMBL8086913 1.00 KMT2A (1.00) KMT2APDE4AMEN1CHRM1PDE4D
Dextofisopam SCHEMBL29376877 1.00 KMT2A (1.00) KMT2APDE4AMEN1CHRM1PDE4D
Tofisopam SCHEMBL4585183 1.00 KMT2A (1.00) KMT2APDE4AMEN1CHRM1PDE4D
Tofisopam SCHEMBL8086894 1.00 KMT2A (1.00) KMT2APDE4AMEN1CHRM1PDE4D
SCHEMBL5426026 0.94 PDE4A (0.88) KMT2APDE4AMEN1CHRM1PDE4D
SCHEMBL5424919 0.94 PDE4A (0.88) KMT2APDE4AMEN1CHRM1PDE4D
SCHEMBL5425481 0.94 PDE4A (0.88) KMT2APDE4AMEN1CHRM1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4547 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12629363-B2 Prophylaxis and treatment of angioedema PHARVARIS GMBH (CH) 2026-05-19 US claimed
EP-3507371-B1 COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM UNIV RUTGERS (US) 2026-01-28 EP claimed
US-20250275979-A1 TREATMENT OF HAIR LOSS DISORDERS WITH DEUTERATED JAK INHIBITORS SUN PHARMACEUTICAL INDUSTRIES, INC. 2025-09-04 US claimed
US-20250179064-A1 BENZOQUINOLONE INHIBITORS OF VMAT2 AUSPEX PHARMACEUTICALS LLC 2025-06-05 US claimed
WO-2024211746-A1 TREATMENT OF AUTOIMMUNE DISEASES AND CANCER WITH PROTEASE INHIBITORS LUNDQUIST INSTITUTE FOR BIOMEDICAL INNOVATION AT HARBOR-UCLA MEDICAL CENTER (US) 2024-10-10 WO claimed
US-20240325404-A1 TREATMENT OF INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2024-10-03 US claimed
US-20240207233-A1 MEDICAMENT KOWA COMPANY, LTD. (JP) 2024-06-27 US claimed
EP-3851541-B1 METHOD FOR RECOVERING TWO OR MORE GENES, OR GENE PRODUCTS, ENCODING AN IMMUNORECEPTOR MEMO THERAPEUTICS AG (CH) 2024-06-05 EP claimed
EP-4370128-A1 TREATMENT OF INFLAMMATORY DISEASES Galapagos N.V. (BE) 2024-05-22 EP claimed
EP-3488338-B1 TECHNOLOGIES FOR ADAPTIVE PROCESSING OF MULTIPLE BUFFERS INTEL CORP (US) 2024-04-17 EP claimed
EP-0117832-B1 VEHICLE MULTIPLEX SYSTEM HAVING PROTOCOL/FORMAT FOR SECURE COMMUNICATION TRANSACTIONS ESSEX GROUP INC. (US) 1988-11-17 EP claimed
EP-0066605-B1 CHIP TOPOGRAPHY FOR INTEGRATED CIRCUIT COMMUNICATION CONTROLLER NCR CORPORATION (US) 1988-11-02 EP claimed
EP-0126384-B1 METHOD AND ARRANGEMENT FOR DECODING AN NB/(N+1)B-CODED DATA STREAM SIEMENS AKTIENGESELLSCHAFT (DE) 1988-10-19 EP claimed
EP-0149766-B1 DEVICE FOR BUILDING UP A FRAME AT THE TRANSMITTING TERMINAL OR DECOMPOSING THE FRAME AT THE RECEIVING TERMINAL RESPECTIVELY FOR A DIGITAL DIRECTIONAL LINK ANT Nachrichtentechnik GmbH (DE) 1988-06-29 EP claimed
EP-0036483-B1 INFORMATION TRANSFER BETWEEN A MAIN STORAGE AND A CYCLIC BULK MEMORY IN A DATA PROCESSING SYSTEM International Business Machines Corporation (US) 1987-02-04 EP claimed
EP-0121658-B1 MEASUREMENT DEVICE Dr. Johannes Heidenhain GmbH (DE) 1986-12-03 EP claimed
EP-0058011-B1 WORD PROCESSING SYSTEM Syntrex Incorporated (US) 1986-11-26 EP claimed
EP-0066532-B1 ELECTRONIC CONTROL APPARATUS SIEMENS AKTIENGESELLSCHAFT (DE) 1986-08-06 EP claimed
EP-0039796-B1 CONTROL CIRCUIT FOR A WRITE HEAD WITH ELECTRODES ARRANGED IN AN INCLINED LINE OF A METALLIZED-PAPER PRINTER IBM DEUTSCHLAND GMBH (DE) 1985-07-31 EP claimed
US-RE30014-E 1-(3,4-Dimethoxy-phenyl)-4-methyl-5-ethyl-7,8-dimethoxy-5H-2,3-benzodiazepine Egyesult Gyogyazer-es Tapozergyar (HU) 1979-05-29 US claimed