SCHEMBL4354019

SCHEMBL4354019

O=C(NCc1ccc(C(F)(F)F)cc1)N(S)c1ccc(O)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.45
HDAC3 O15379 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
MTOR P42345 2/20 0.43
LSS P48449 1/20 0.43
MAPK14 Q16539 1/20 0.41
DUSP3 P51452 1/20 0.41
KCNH2 Q12809 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39
ESRRG P62508 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
KDM1A O60341 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4341863 0.89 HDAC3 (0.48) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL4357663 0.87 HDAC1 (0.44) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL4341578 0.83 POLB (0.43) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL4342201 0.81 EPHX2 (0.45) MTORTRPV1CA12CA1CA2
SCHEMBL4357500 0.80 HDAC3 (0.46) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL4351640 0.80 HDAC1 (0.49) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL4359745 0.78 TMPRSS4 (0.50) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL3298777 0.78 CCR2 (0.47) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL4348897 0.77 MTOR (0.50) HDAC1HDAC3HDAC2HDAC10HDAC11
SCHEMBL4354458 0.77 MTOR (0.42) HDAC1HDAC3HDAC2HDAC10HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed