SCHEMBL4354244

SCHEMBL4354244

COC(=O)c1c(Nc2ccc(F)cc2)cnn1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BPTF Q12830 3/20 0.56
PDE10A Q9Y233 1/20 0.51
CNR2 P34972 1/20 0.46
MAPK14 Q16539 1/20 0.44
TP53 P04637 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
GAA P10253 1/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HTR2C P28335 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTR2A P28223 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6785353 0.86 BPTF (0.58) BPTFPDE10AKMT2AMEN1GAA
SCHEMBL4354248 0.81 CYP1A2 (0.54) PDE10ACNR2NPC1RAB9AMAPT
SCHEMBL24485756 0.74 CNR2 (0.46) CNR2TP53KMT2AMEN1HTT
SCHEMBL30908549 0.73 CNR2 (0.59) PDE10ACNR2MAPTKMT2AMEN1
SCHEMBL6786160 0.72 BPTF (0.44) BPTFPDE10ANPC1RAB9AMAPT
SCHEMBL6789292 0.71 SMN1; SMN2 (0.48) BPTFPDE10ANPC1RAB9AMAPT
SCHEMBL18255876 0.71 CNR2 (0.54) PDE10ACNR2KMT2AMEN1HTT
SCHEMBL26910162 0.71 BPTF (1.00) BPTF
SCHEMBL8834288 0.71 MAPT (0.51) NPC1RAB9AMAPTKMT2AMEN1
SCHEMBL27409311 0.71 CNR2 (0.56) PDE10ACNR2KMT2AMEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026241-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2009-02-26 WO disclosed