SCHEMBL4354885

SCHEMBL4354885

CCCc1n[nH]c(=O)c(C(=O)OCC)c1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.47
ADORA1 P30542 1/20 0.47
PDE1A P54750 1/20 0.47
PDE1B Q01064 1/20 0.47
PDE3B Q13370 1/20 0.47
PDE1C Q14123 1/20 0.47
PDE3A Q14432 1/20 0.47
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
LMNA P02545 1/20 0.44
KDM5A P29375 1/20 0.43
KDM5B Q9UGL1 1/20 0.43
APLNR P35414 1/20 0.43
POLB P06746 1/20 0.43
KDM4E B2RXH2 2/20 0.42
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4574454 0.84 PDE4D (0.46) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL3849702 0.83 PDE4D (0.64) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL14006504 0.81 ADORA1 (0.44) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL3853102 0.80 POLB (0.56) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL3846991 0.77 PDE4D (0.47) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL3855819 0.77 PDE4D (0.47) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL21585140 0.76 PDE4D (0.50) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL3848316 0.75 KDM4E (0.52) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL20338259 0.74 PDE4D (0.66) PDE4DADORA1PDE1APDE1BPDE3B
SCHEMBL3847496 0.72 HPGDS (0.60) ALDH1A1SMN1; SMN2LMNAPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124565-A2 N-SUBSTITUTED GLYCINE DERIVATIVES: HYDROXYLASE INHIBITORS Smithkline Beecham Corporation (US) 2009-12-02 EP disclosed
WO-2008089052-A2 N-SUBSTITUTED GLYCINE DERIVATIVES: HYDROXYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-24 WO disclosed