SCHEMBL4356685

SCHEMBL4356685

O=C(CCc1ccccc1)N[C@H]1CCCN2CCC[C@@H](C(=O)NC3CC(=O)OC3OCc3ccccc3)N2C1=O

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 6/20 0.49
CASP3 P42574 5/20 0.49
CASP8 Q14790 4/20 0.49
ACE P12821 3/20 0.45
MME P08473 2/20 0.45
KLK7 P49862 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL647366 1.00 CASP1 (0.49) CASP1CASP3CASP8ACEMME
SCHEMBL1409861 1.00 CASP1 (0.49) CASP1CASP3CASP8ACEMME
SCHEMBL644997 0.90 CASP1 (0.60) CASP1CASP3CASP8ACEMME
SCHEMBL1414605 0.90 CASP1 (0.60) CASP1CASP3CASP8ACEMME
SCHEMBL1409707 0.90 CASP1 (0.60) CASP1CASP3CASP8ACEMME
SCHEMBL644933 0.89 CASP1 (0.52) CASP1CASP3CASP8ACEMME
SCHEMBL644714 0.89 CASP1 (0.52) CASP1CASP3CASP8ACEMME
SCHEMBL1414638 0.89 CASP1 (0.52) CASP1CASP3CASP8ACEMME
SCHEMBL1410174 0.89 CASP1 (0.52) CASP1CASP3CASP8ACEMME
SCHEMBL12450751 0.89 CASP1 (0.52) CASP1CASP3CASP8ACEMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083014-A2 Inhibitors of interleukin-1ß converting enzyme Vertex Pharmceuticals Incorporated (US) 2009-07-29 EP disclosed
US-6258948-B1 AN N-ACYLAMINO COMPOUND; ANTIINFLAMMATORY AGENTS, AUTOIMMUNE DISEASES VERTEX PHARMACEUTICALS, INCORPORATED 2001-07-10 US disclosed