SCHEMBL4356795

SCHEMBL4356795

CN(C)C1CCCN(C(=O)C2COCCN2C(=O)c2cc3ccccc3[nH]2)C1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
AKR1C3 P42330 9/20 0.47
HRH4 Q9H3N8 5/20 0.45
HRH3 Q9Y5N1 1/20 0.41
F2 P00734 1/20 0.41
F10 P00742 1/20 0.41
PLG P00747 1/20 0.41
PRSS1 P07477 1/20 0.41
RBP4 P02753 1/20 0.40
PDE4B Q07343 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4361046 0.78 PROKR1 (0.43)
SCHEMBL4327043 0.77 HRH4 (0.63) POLBSMN1; SMN2AKR1C3HRH4HRH3
SCHEMBL3540795 0.74 POLB (0.51) POLBSMN1; SMN2AKR1C3HRH4HRH3
SCHEMBL2347853 0.73 POLB (0.63) POLBSMN1; SMN2AKR1C3HRH4HRH3
SCHEMBL24235367 0.71 AKR1C3 (0.61) POLBSMN1; SMN2AKR1C3HRH4HRH3
SCHEMBL30310614 0.70 AKR1C3 (0.60) POLBSMN1; SMN2AKR1C3HRH4HRH3
SCHEMBL13753537 0.69 AKR1C3 (0.62) POLBSMN1; SMN2AKR1C3HRH4HRH3
SCHEMBL15064997 0.69 AKR1C3 (0.62) POLBSMN1; SMN2AKR1C3HRH4HRH3
SCHEMBL28551515 0.69 KDM4E (0.44) POLBSMN1; SMN2AKR1C3HRH4
SCHEMBL25040621 0.69 HRH4 (0.64) AKR1C3HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010487-A1 5-AMIDO-2-CARBOXAMIDE INDOLES F. Hoffmann-Roche AG (CH) 2009-01-07 EP disclosed
WO-2007115938-A1 5-AMIDO-2-CARBOXAMIDE INDOLES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-18 WO disclosed