SCHEMBL4366311

SCHEMBL4366311

CC(C)C[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)C(=O)N1CC[C@@H]2C1C(=O)CN2C(=O)OC(C)(C)C

nearest known ligand 0.77

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.77
CTSS P25774 1/20 0.57
MAPK1 P28482 2/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CCR1 P32246 1/20 0.39
POLB P06746 2/20 0.38
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5941473 1.00 CTSK (0.77) CTSKCTSSMAPK1ALDH1A1LMNA
SCHEMBL4048050 0.90 CTSK (0.75) CTSKCTSSCCR1POLB
SCHEMBL4041814 0.89 CTSK (0.79) CTSKCTSSALDH1A1MEN1KMT2A
SCHEMBL4039416 0.88 CTSK (0.78) CTSKCTSSALDH1A1MEN1KMT2A
SCHEMBL4041202 0.88 CTSK (0.80) CTSKCTSSCCR1POLB
SCHEMBL4040161 0.88 CTSK (0.74) CTSKCTSSCCR1POLB
SCHEMBL4224757 0.88 CTSK (0.77) CTSKCTSSALDH1A1MEN1KMT2A
SCHEMBL4038929 0.88 CTSK (0.77) CTSKCTSSALDH1A1MEN1KMT2A
SCHEMBL4042931 0.88 CTSK (0.77) CTSKCTSSCCR1
SCHEMBL4048538 0.88 CTSK (0.77) CTSKCTSSALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP disclosed