SCHEMBL436633

SCHEMBL436633

Nc1c(C(=O)O)cnc2c(F)cccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.68
ALB P02768 1/20 0.42
AURKA O14965 2/20 0.42
RAB9A P51151 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
PARP1 P09874 1/20 0.41
NR1H2 P55055 2/20 0.40
NR1H3 Q13133 2/20 0.40
KDM4E B2RXH2 3/20 0.40
KDM4A O75164 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40
HIF1AN Q9NWT6 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
BTK Q06187 1/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
G6PD P11413 1/20 0.39
CASP7 P55210 1/20 0.39
CASP6 P55212 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6198659 0.83 ALB (0.51) HAVCR2ALBAURKARAB9AKMT2A
SCHEMBL2719152 0.81 HAVCR2 (0.52) HAVCR2ALBAURKARAB9AKMT2A
SCHEMBL436943 0.81 HAVCR2 (0.56) HAVCR2RAB9AKMT2ANPC1KDM4E
SCHEMBL436434 0.81 HAVCR2 (0.68) HAVCR2RAB9AKMT2ANPC1KDM4E
SCHEMBL10126289 0.81 HAVCR2 (0.68) HAVCR2AURKAPARP1BTKG6PD
SCHEMBL436716 0.81 HAVCR2 (1.00) HAVCR2AURKARAB9AKMT2ANPC1
SCHEMBL437026 0.81 HAVCR2 (0.68) HAVCR2AURKARAB9AKMT2ANPC1
SCHEMBL440043 0.79 KMT2A (0.68) RAB9AKMT2ANPC1KDM4EMAPK1
SCHEMBL26167923 0.79 HAVCR2 (0.54) HAVCR2AURKARAB9AKMT2ANPC1
SCHEMBL442207 0.79 HAVCR2 (0.65) HAVCR2RAB9AKMT2ANPC1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed