SCHEMBL4366407

SCHEMBL4366407

O=C(O)c1ccc2[nH]c(-c3nc4ccc(C(=O)O)cc4[nH]3)nc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.65
CHEK2 O96017 9/20 0.63
HSP90AA1 P07900 1/20 0.62
ESR2 Q92731 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
SMN1; SMN2 Q16637 2/20 0.57
NPSR1 Q6W5P4 1/20 0.57
MMP2 P08253 1/20 0.57
MMP9 P14780 1/20 0.57
MMP8 P22894 1/20 0.57
MMP13 P45452 1/20 0.57
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 2/20 0.55
HPGD P15428 2/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
APEX1 P27695 1/20 0.55
KMT2A Q03164 1/20 0.54
F2 P00734 1/20 0.52
F10 P00742 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL828113 0.93 KDM4E (0.56) NR4A2CHEK2HSP90AA1ESR2TDP1
SCHEMBL20982594 0.92 NR4A2 (0.77) NR4A2CHEK2SMN1; SMN2MMP2MMP9
SCHEMBL28930292 0.85 KDM4E (0.68) NR4A2CHEK2SMN1; SMN2MMP2MMP9
SCHEMBL20982644 0.85 NR4A2 (0.86) NR4A2CHEK2HSP90AA1ESR2TDP1
SCHEMBL7602620 0.84 KDM4E (0.70) NR4A2CHEK2SMN1; SMN2MMP2MMP9
SCHEMBL5219768 0.84 NR4A2 (0.83) NR4A2CHEK2MMP2MMP9MMP8
SCHEMBL3178116 0.83 CHEK2 (0.78) NR4A2CHEK2SMN1; SMN2MMP2MMP9
SCHEMBL28722299 0.83 NR4A2 (0.72) NR4A2CHEK2HSP90AA1ESR2TDP1
SCHEMBL8611783 0.83 KDM4E (0.69) NR4A2CHEK2SMN1; SMN2MMP2MMP9
SCHEMBL28722301 0.83 KDM4E (0.61) NR4A2CHEK2HSP90AA1ESR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081913-A2 BENZIMIDAZOLE,BENZOXAZOLE AND BENZOTHIAZOLE DERIVATIVES, OPTICAL FILM COMPRISING THEM AND METHOD OF PRODUCTION THEREOF CRYSOPTIX K.K. (JP) 2009-07-29 EP disclosed
WO-2008020211-A2 BENZIMIDAZOLE, BENZOXAZOLE AND BENZOTHIAZOLE DERIVATIVES, OPTICAL FILM COMPRISING THEM AND METHOD OF PRODUCTION THEREOF CRYSOPTIX K.K. (JP) 2008-02-21 WO disclosed