SCHEMBL4367186

SCHEMBL4367186

CC(C)(C)OC(=O)N1CCC[C@@H]1COc1cc(N)ccc1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 3/20 0.48
FEN1 P39748 1/20 0.48
UTS2R Q9UKP6 2/20 0.42
WNT3 P56703 2/20 0.41
SFRP1 Q8N474 2/20 0.41
F2RL3 Q96RI0 4/20 0.41
NR1H2 P55055 1/20 0.40
GPR119 Q8TDV5 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4372549 1.00 ALOX5AP (0.48) ALOX5APFEN1UTS2RWNT3SFRP1
SCHEMBL449546 0.92 ALOX5AP (0.47) ALOX5APFEN1F2RL3NR1H2GPR119
SCHEMBL447304 0.92 ALOX5AP (0.47) ALOX5APFEN1F2RL3NR1H2GPR119
SCHEMBL447303 0.92 ALOX5AP (0.47) ALOX5APFEN1F2RL3NR1H2GPR119
SCHEMBL448827 0.92 ALOX5AP (0.47) ALOX5APFEN1F2RL3NR1H2GPR119
SCHEMBL448828 0.92 ALOX5AP (0.47) ALOX5APFEN1F2RL3NR1H2GPR119
SCHEMBL520556 0.86 ALOX5AP (0.47) ALOX5APFEN1F2RL3NR1H2GPR119
SCHEMBL521653 0.86 ALOX5AP (0.47) ALOX5APFEN1F2RL3NR1H2GPR119
SCHEMBL13419700 0.86 ALOX5AP (0.51) ALOX5APFEN1F2RL3NR1H2GPR119
SCHEMBL520557 0.86 ALOX5AP (0.47) ALOX5APFEN1F2RL3NR1H2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed
EP-1638954-A1 FUSED AZOLES SUCH AS 2,5-DISUBSTITUTED BENZIMIDAZOLES, BENZOXAZOLES AND BENZOTHIAZOLES AS KINASE INHIBITORS AMGEN INC. (US) 2006-03-29 EP disclosed
US-20040209892-A1 Heterocyclic compounds and methods of use U.S. PATENT OPERATIONS 2004-10-21 US disclosed
WO-2004085425-A1 FUSED AZOLES SUCH AS 2,5-DISUBSTITUTED BENZIMIDAZOLES, BENZOXAZOLES AND BENZOTHIAZOLES AS KINASE INHIBITORS AMGEN INC (US) 2004-10-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209892-A1 Heterocyclic compounds and methods of use VHL, NQO1, HPGDS ALOX5AP 555/4885FEN1 1212/4885UTS2R 2684/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.