SCHEMBL436978

SCHEMBL436978

Fc1c[c]ccc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.40
HSD11B1 P28845 2/20 0.38
KDM4E B2RXH2 3/20 0.36
TP53 P04637 2/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 2/20 0.33
IDO1 P14902 1/20 0.33
AQP1 P29972 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
CRHR1 P34998 1/20 0.33
MAPT P10636 1/20 0.33
CYP3A4 P08684 2/20 0.32
TSHR P16473 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433088 0.89 KMO (0.36) AHRHSD11B1
SCHEMBL432656 0.86 KMO (0.35) AHRHSD11B1KDM4ETP53RAB9A
SCHEMBL17514770 0.86 NISCH (0.38) HSD11B1KDM4ETP53RAB9ANPC1
SCHEMBL435070 0.85 AHR (0.45) AHRHSD11B1KDM4ETP53RAB9A
SCHEMBL1984033 0.79 AHR (0.44) AHRHSD11B1KDM4ETP53RAB9A
SCHEMBL27688592 0.79 KMO (0.35) AHRHSD11B1KDM4ETP53RAB9A
SCHEMBL16720300 0.79 HSD17B10 (0.45) AHRHSD11B1KDM4ETP53SMN1; SMN2
SCHEMBL2886283 0.78
SCHEMBL7822011 0.78 CYP2A6 (0.39) HSD11B1TP53RAB9ANPC1SMN1; SMN2
SCHEMBL27707557 0.76 KMO (0.36) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed