SCHEMBL4369908

SCHEMBL4369908

Fc1ccc(Nc2nc3cc(Oc4ccncc4)ccc3[nH]2)cc1F

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.56
PDE10A Q9Y233 6/20 0.44
RAF1 P04049 8/20 0.43
CSNK1A1 P48729 2/20 0.42
CSNK1D P48730 2/20 0.42
BRAF P15056 7/20 0.42
HDAC11 Q96DB2 1/20 0.39
GSK3B P49841 1/20 0.39
CSNK1G2 P78368 1/20 0.39
TEK Q02763 1/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4364072 0.90 KDR (0.61) KDRPDE10ARAF1CSNK1A1CSNK1D
SCHEMBL4367856 0.88 KDR (0.55) KDRPDE10ARAF1CSNK1A1CSNK1D
SCHEMBL4375547 0.85 KDR (0.53) KDRPDE10ARAF1CSNK1A1CSNK1D
SCHEMBL13861947 0.84 KDR (0.61) KDRPDE10ARAF1CSNK1A1CSNK1D
SCHEMBL4369261 0.83 CSNK1A1 (0.54) KDRPDE10ARAF1CSNK1A1CSNK1D
SCHEMBL4370234 0.83 KDR (0.55) KDRPDE10ARAF1CSNK1A1CSNK1D
SCHEMBL4161669 0.82 KDR (0.56) KDRPDE10ARAF1CSNK1A1CSNK1D
SCHEMBL2893930 0.81 RAF1 (0.67) KDRRAF1BRAF
SCHEMBL4372559 0.81 KDR (0.85) KDRPDE10ARAF1CSNK1A1CSNK1D
SCHEMBL13862513 0.81 KDR (0.61) KDRPDE10ARAF1CSNK1A1CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed
US-20040209892-A1 Heterocyclic compounds and methods of use U.S. PATENT OPERATIONS 2004-10-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209892-A1 Heterocyclic compounds and methods of use VHL, NQO1, HPGDS KDR 83/4885PDE10A 947/4885RAF1 1846/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.