SCHEMBL4371052

SCHEMBL4371052

CC(C)C[C@H](NC(=O)c1cccc(Oc2ccccc2)c1)C(=O)N1CCC2[C@H]1C(=O)CN2C(=O)c1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSK P43235 9/20 0.72
CTSS P25774 5/20 0.54
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CCR1 P32246 1/20 0.43
CTSL P07711 5/20 0.42
NPC1 O15118 1/20 0.41
CFTR P13569 1/20 0.40
CTSV O60911 2/20 0.40
PKM P14618 1/20 0.40
CCKBR P32239 1/20 0.39
GPR139 Q6DWJ6 1/20 0.39
CTSB P07858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4371066 1.00 CTSK (0.72) CTSKCTSSALDH1A1LMNASMN1; SMN2
SCHEMBL4371059 1.00 CTSK (0.72) CTSKCTSSALDH1A1LMNASMN1; SMN2
SCHEMBL5942128 1.00 CTSK (0.72) CTSKCTSSALDH1A1LMNASMN1; SMN2
SCHEMBL4375538 0.93 CTSK (0.80) CTSKCTSSCCR1CTSLCTSV
SCHEMBL4375532 0.93 CTSK (0.80) CTSKCTSSCCR1CTSLCTSV
SCHEMBL5941645 0.93 CTSK (0.80) CTSKCTSSCCR1CTSLCTSV
SCHEMBL4375530 0.93 CTSK (0.80) CTSKCTSSCCR1CTSLCTSV
SCHEMBL5942142 0.92 CTSK (0.62) CTSKCTSSALDH1A1LMNASMN1; SMN2
SCHEMBL5942144 0.92 CTSK (0.62) CTSKCTSSALDH1A1LMNASMN1; SMN2
SCHEMBL5941948 0.92 CTSK (0.82) CTSKCTSSALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP disclosed