SCHEMBL4372271

SCHEMBL4372271

COc1ccc2c(c1OC)CC=C(C)[CH]2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
HPGD P15428 2/20 0.40
ACHE P22303 3/20 0.37
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33
TUBB2A Q13885 1/20 0.33
TUBB8 Q3ZCM7 1/20 0.33
TUBA3E Q6PEY2 1/20 0.33
TUBA1A Q71U36 1/20 0.33
TUBA1C Q9BQE3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4308679 0.71 KDM4E (0.42) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL4310800 0.70 KMT2A (0.39) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL3674074 0.65 CA9 (0.50) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL30701949 0.65 CA9 (0.50) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL10681803 0.64 KDM4E (0.46) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL27914001 0.63 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL9573206 0.62 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL27996930 0.62 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL11591320 0.62 KDM4E (0.40) ALDH1A1KDM4EHPGDACHECA1
SCHEMBL3158365 0.62 KDM4E (0.56) ALDH1A1KDM4EHPGDACHEGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117601-A2 MACROMOLECULAR CONJUGATES OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR PROTEIN INHIBITORS AND USES THEREOF The Regents of the University of California (US) 2009-11-18 EP disclosed
WO-2008079897-A2 MACROMOLECULAR CONJUGATES OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR PROTEIN INHIBITORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2008-07-03 WO disclosed