SCHEMBL4373330

SCHEMBL4373330

COc1ccccc1COc1ccc(-c2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)NCc3ccccc3)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.54
MMP2 P08253 4/20 0.53
KLKB1 P03952 1/20 0.52
HTT P42858 1/20 0.51
NFKB1 P19838 1/20 0.49
PSMB5 P28074 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
ADAMTS5 Q9UNA0 2/20 0.48
MMP8 P22894 1/20 0.48
MMP12 P39900 1/20 0.48
ADAMTS4 O75173 1/20 0.48
KDM1A O60341 2/20 0.47
HPGD P15428 1/20 0.46
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
HDAC3 O15379 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3588838 0.88 FFAR1 (0.53) KLKB1NFKB1PSMB5NFKB2RELA
SCHEMBL3588585 0.88 KLKB1 (0.57) MMP2KLKB1NFKB1PSMB5NFKB2
SCHEMBL2246373 0.87 HTT (0.67) MMP2HTTADAMTS5MMP8MMP12
SCHEMBL3589157 0.87 KLKB1 (0.50) MMP2KLKB1NFKB1PSMB5NFKB2
SCHEMBL3583762 0.87 CTSS (0.53) MMP2KLKB1HTTNFKB1PSMB5
SCHEMBL3583723 0.86 KLKB1 (0.54) MMP2KLKB1NPC1RAB9AADAMTS5
SCHEMBL3584887 0.85 KLKB1 (0.69) MMP2KLKB1L3MBTL1NPC1RAB9A
SCHEMBL2251666 0.85 NPC1 (0.67) MMP2KLKB1NPC1RAB9AADAMTS5
SCHEMBL3595965 0.84 KLKB1 (0.53) MMP2KLKB1NPC1RAB9AADAMTS5
SCHEMBL3577147 0.84 KLKB1 (0.56) MMP2KLKB1HTTNFKB1PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553873-B2 Glutamate aggrecanase inhibitors WYETH (US) 2009-06-30 US claimed