SCHEMBL4373986

SCHEMBL4373986

CN(CCN(CCC12CC3CC(CC(C3)C1)C2)C(=O)NCCCc1cc[n+](C)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 10/20 0.35
EPHX1 P07099 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
FPR3 P25089 1/20 0.34
FPR2 P25090 1/20 0.34
HDAC11 Q96DB2 1/20 0.33
CXCR3 P49682 1/20 0.33
P2RX7 Q99572 3/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CASP2 P42575 1/20 0.31
ABCB11 O95342 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL1677836 0.99 EPHX2 (0.35) EPHX2EPHX1ALDH1A1SMN1; SMN2FPR3
SCHEMBL1677543 0.89 P2RX7 (0.39) EPHX2EPHX1ALDH1A1SMN1; SMN2FPR3
SCHEMBL1678508 0.85 P2RX7 (0.39) EPHX2EPHX1ALDH1A1SMN1; SMN2FPR3
SCHEMBL1677528 0.85 P2RX7 (0.39) EPHX2EPHX1ALDH1A1SMN1; SMN2FPR3
SCHEMBL1678221 0.82 P2RX7 (0.38) EPHX2EPHX1ALDH1A1SMN1; SMN2HDAC11
Iodide SCHEMBL1677581 0.81 EPHX2 (0.40) EPHX2EPHX1ALDH1A1SMN1; SMN2P2RX7
SCHEMBL1678145 0.81 P2RX7 (0.37) EPHX2EPHX1ALDH1A1SMN1; SMN2HDAC11
SCHEMBL1678526 0.80 NAMPT (0.42) EPHX2EPHX1ALDH1A1SMN1; SMN2P2RX7
SCHEMBL1679354 0.80 P2RX7 (0.42) EPHX2EPHX1ALDH1A1SMN1; SMN2HDAC11
SCHEMBL1677680 0.78 P2RX7 (0.40) EPHX2EPHX1ALDH1A1SMN1; SMN2HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1743885-B1 1-[(adamantyl)alkyl]-3-[(pyridinyl)alkyl]urea compounds as TNF-.alpha inhibitors useful for autoimmune diseases SANTEN PHARMACEUTICAL CO LTD (JP) 2009-11-11 EP disclosed
EP-1743885-A2 TNF-Alpha Produktion Hemmer zur Behandlung von Autoimmunerkrankungen SANTEN PHARMACEUTICAL CO., LTD. (JP) 2007-01-17 EP disclosed