SCHEMBL4374093

SCHEMBL4374093

Cc1nn(-c2ccc(C#N)c(N)c2)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 17/20 0.60
HSP90AB1 P08238 3/20 0.59
HSP90AA1 P07900 2/20 0.52
OPRK1 P41145 3/20 0.50
OPRD1 P41143 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16883487 0.89 OPRM1 (0.62) OPRM1HSP90AB1OPRK1OPRD1
SCHEMBL3632840 0.87 OPRM1 (0.60) OPRM1HSP90AB1HSP90AA1OPRK1OPRD1
SCHEMBL27649673 0.87 OPRM1 (0.66) OPRM1HSP90AB1OPRK1OPRD1
SCHEMBL1219080 0.87 OPRM1 (0.66) OPRM1HSP90AB1HSP90AA1OPRK1OPRD1
SCHEMBL12191669 0.87 OPRM1 (0.60) OPRM1HSP90AB1HSP90AA1OPRK1OPRD1
SCHEMBL2775193 0.85 HSP90AB1 (0.66) OPRM1HSP90AB1HSP90AA1OPRK1OPRD1
SCHEMBL21558179 0.82 OPRM1 (0.65) OPRM1HSP90AB1HSP90AA1OPRK1OPRD1
SCHEMBL28761859 0.82 HSP90AB1 (0.55) OPRM1HSP90AB1HSP90AA1OPRK1OPRD1
SCHEMBL3627830 0.81 OPRM1 (0.58) OPRM1HSP90AB1OPRK1OPRD1
SCHEMBL4369836 0.81 HSP90AB1 (0.56) OPRM1HSP90AB1HSP90AA1OPRK1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009114470-A2 TETRAHYDROINDOLE AND TETRAHDYROINDAZOLE AS HSP90 INHIBITORS CONTAINING A ZINC BINDING MOIETY CURIS, INC. (US) 2009-09-17 WO disclosed
WO-2009114470-A2 TETRAHYDROINDOLE AND TETRAHDYROINDAZOLE AS HSP90 INHIBITORS CONTAINING A ZINC BINDING MOIETY CURIS, INC. (US) 2009-09-17 WO disclosed