SCHEMBL4375574

SCHEMBL4375574

COc1cc2c(Cl)ncnc2cc1OCCCN(C)S(C)(=O)=O

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 6/20 0.62
EGFR P00533 5/20 0.47
KDR P35968 8/20 0.45
CSF1R P07333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16760479 0.94 ENPP1 (0.64) ENPP1EGFRKDRCSF1R
SCHEMBL3947513 0.86 ENPP1 (0.71) ENPP1EGFRKDRCSF1R
SCHEMBL1012226 0.83 ENPP1 (0.68) ENPP1KDR
SCHEMBL4373124 0.83 ENPP1 (0.68) ENPP1KDR
SCHEMBL1011386 0.82 ENPP1 (0.70) ENPP1KDR
SCHEMBL3951030 0.82 ENPP1 (0.73) ENPP1EGFRKDRCSF1R
SCHEMBL1015576 0.80 ENPP1 (0.79) ENPP1EGFRKDRCSF1R
SCHEMBL1013051 0.80 ENPP1 (0.79) ENPP1EGFRKDRCSF1R
SCHEMBL30864338 0.80 ENPP1 (0.79) ENPP1EGFRKDRCSF1R
SCHEMBL31620798 0.80 ENPP1 (0.79) ENPP1EGFRKDRCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8492560-B2 Quinazoline derivatives as angiogenesis inhibitors ASTRAZENECA AB (SE) 2013-07-23 US disclosed
US-20120197027-A1 Quinazoline Derivatives as Angiogenesis Inhibitors STOKES ELAINE S E (GB) 2012-08-02 US disclosed
EP-2050744-A1 Quinazoline derivatives as angiogenesis inhibitors AstraZeneca AB (SE) 2009-04-22 EP disclosed
US-7074800-B1 Quinazoline derivatives as angiogenesis inhibitors ASTRAZENECA AB (SE) 2006-07-11 US disclosed
EP-1553097-A1 QUINAZOLINE DERIVATIVES AS ANGIOGENESIS INHIBITORS AND INTERMEDIATES THEREFORE AstraZeneca AB (SE) 2005-07-13 EP disclosed
EP-1154774-A1 QUINAZOLINE DERIVATIVES AS ANGIOGENESIS INHIBITORS AstraZeneca AB (SE) 2001-11-21 EP disclosed
WO-2000047212-A1 QUINAZOLINE DERIVATIVES AS ANGIOGENESIS INHIBITORS ASTRAZENECA AB (SE) 2000-08-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120197027-A1 Quinazoline Derivatives as Angiogenesis Inhibitors VEGFA, FLT1, KDR ENPP1 2575/4885EGFR 500/4885KDR 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.