Flumizole

Flumizole

SCHEMBL43779

COc1ccc(-c2nc(C(F)(F)F)[nH]c2-c2ccc(OC)cc2)cc1

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.58
ESR2 Q92731 1/20 0.58
NOX1 Q9Y5S8 1/20 0.55
MAPK13 O15264 2/20 0.52
MAPK12 P53778 2/20 0.52
MAPK11 Q15759 2/20 0.52
MAPK14 Q16539 2/20 0.52
ALOX5 P09917 1/20 0.52
GCGR P47871 1/20 0.52
MAPT P10636 5/20 0.50
TP53 P04637 2/20 0.50
SMPD3 Q9NY59 1/20 0.50
PDE10A Q9Y233 1/20 0.50
RAF1 P04049 1/20 0.50
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
LMNA P02545 2/20 0.48
HTT P42858 2/20 0.48
TDP1 Q9NUW8 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flumizole SCHEMBL15757137 1.00 ESR1 (0.58) ESR1ESR2NOX1MAPK13MAPK12
SCHEMBL7089213 0.91 ESR1 (0.50) ESR1ESR2NOX1MAPK13MAPK12
SCHEMBL7087514 0.88 TEK (0.53) ESR1ESR2MAPK11MAPK14ALOX5
SCHEMBL7089441 0.87 PTGS1 (0.50) ESR1ESR2NOX1ALOX5
SCHEMBL11164692 0.85 NOX1 (0.50) ESR1ESR2NOX1MAPK13MAPK12
SCHEMBL11087790 0.85 NOX1 (0.50) ESR1ESR2NOX1MAPK13MAPK12
SCHEMBL11165161 0.85 NOX1 (0.53) ESR1ESR2NOX1MAPK13MAPK12
SCHEMBL11177941 0.84 NOX1 (0.52) ESR1ESR2NOX1MAPK13MAPK12
SCHEMBL11170006 0.83 NOX1 (0.57) ESR1ESR2NOX1MAPK13MAPK12
SCHEMBL11177151 0.82 NOX1 (0.50) ESR1ESR2NOX1MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3564 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ACERAGEN INC (US) 2026-01-01 US claimed
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
WO-2023212179-A2 THERAPEUTIC COMPOSITIONS FOR SKIN DISORDERS AND WOUND REPAIR UNIVERSITY OF MIAMI (US) 2023-11-02 WO claimed
US-20220110979-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC 2022-04-14 US claimed
US-20220088158-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ROIVANT SCIENCES, INC. 2022-03-24 US claimed
EP-3908297-A1 FIBROBLAST REGENERATIVE CELLS Figene, LLC (US) 2021-11-17 EP claimed
EP-3279663-B1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES BRIGHAM & WOMENS HOSPITAL INC (US) 2021-07-28 EP claimed
WO-2020152532-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ENZYVANT THERAPEUTICS GMBH (CH) 2020-07-30 WO claimed
WO-2020146874-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC (US) 2020-07-16 WO claimed
CN-109860675-A A kind of new-energy automobile fuel cell ion exchange membrane and preparation method thereof 杨记周 2019-06-07 CN claimed
EP-0644755-B1 SURFACE MODIFIED NSAID NANOPARTICLES NANOSYSTEMS LLC (US) 1997-03-19 EP claimed
EP-0759750-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO, Howard, K. (US) 1997-03-05 EP claimed
US-5591456-A ADSORPTION ON HYDROXYPROPYL CELLULOSE NANOSYSTEMS L.L.C. (US) 1997-01-07 US claimed
US-5552160-A NONSTEROID ANALGESICS FOR REDUCED GASTRIC IRRITATION NANOSYSTEMS L.L.C. (US) 1996-09-03 US claimed
WO-1996024336-A1 NSAID NANOPARTICLES NANOSYSTEMS L.L.C. (US) 1996-08-15 WO claimed
WO-1996024339-A1 COMPOSITIONS COMPRISING NANOPARTICLES OF NSAID NANOSYSTEMS L.L.C. (US) 1996-08-15 WO claimed
US-5518738-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS, REDUCED GASTRIC IRRITATION NANOSYSTEM L.L.C. (US) 1996-05-21 US claimed
WO-1995031194-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1995-11-23 WO claimed
EP-0644755-A1 SURFACE MODIFIED NSAID NANOPARTICLES. EASTMAN KODAK CO (US) 1995-03-29 EP claimed
WO-1993025190-A1 SURFACE MODIFIED NSAID NANOPARTICLES EASTMAN KODAK COMPANY (US) 1993-12-23 WO claimed