SCHEMBL4378407

SCHEMBL4378407

NC(=O)C1CN(c2cc(F)c(N3CCCOCC3)c(F)c2)C(=O)O1

nearest known ligand 0.91

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.91
MAOB P27338 10/20 0.44
PTGS1 P23219 2/20 0.44
SDHA P31040 2/20 0.44
LMNA P02545 1/20 0.44
CALML3 P27482 1/20 0.44
F10 P00742 1/20 0.39
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13632911 1.00 MAOA (0.91) MAOAMAOBPTGS1SDHALMNA
SCHEMBL3038122 0.95 MAOA (1.00) MAOAMAOBPTGS1SDHALMNA
SCHEMBL4378718 0.88 MAOA (0.71) MAOAMAOBPTGS1SDHALMNA
SCHEMBL14639627 0.87 MAOA (0.70) MAOAMAOBPTGS1SDHALMNA
SCHEMBL4380781 0.87 MAOA (0.70) MAOAMAOBPTGS1SDHALMNA
SCHEMBL3031991 0.86 MAOA (0.82) MAOAMAOBPTGS1SDHALMNA
SCHEMBL5765718 0.86 MAOA (0.82) MAOAMAOBPTGS1SDHALMNA
SCHEMBL13633151 0.86 MAOA (0.68) MAOAMAOBPTGS1SDHALMNA
SCHEMBL13634014 0.86 MAOA (0.68) MAOAMAOBPTGS1SDHALMNA
SCHEMBL4379493 0.86 MAOA (0.68) MAOAMAOBPTGS1SDHALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899331-B1 HOMOMORPHOLINE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN CO LLC (US) 2009-11-25 EP claimed
EP-1899331-A1 HOMOMORPHOLINE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2008-03-19 EP claimed
WO-2007000644-A1 HOMOMORPHOLINE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2007-01-04 WO claimed
EP-1899331-B1 HOMOMORPHOLINE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN CO LLC (US) 2009-11-25 EP disclosed
EP-1899331-A1 HOMOMORPHOLINE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2008-03-19 EP disclosed
WO-2007000644-A1 HOMOMORPHOLINE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2007-01-04 WO disclosed