SCHEMBL4378709

SCHEMBL4378709

Fc1c(F)c(F)c(-c2ccncc2)c(-c2ccncc2)c1F

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.53
LMNA P02545 2/20 0.53
KDM4E B2RXH2 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
NOTUM Q6P988 1/20 0.43
KIF11 P52732 1/20 0.42
MAPK14 Q16539 12/20 0.41
DDAH1 O94760 1/20 0.39
NOS1 P29475 1/20 0.39
TP53 P04637 1/20 0.39
PKM P14618 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21578111 0.92 MAPT (0.56) MAPTLMNAKDM4ECYP1A2CYP3A4
SCHEMBL21578127 0.82 MAPT (0.46) MAPTLMNAKDM4ECYP1A2CYP3A4
SCHEMBL4302102 0.78 MAPT (0.71) MAPTLMNAKDM4ECYP1A2CYP3A4
SCHEMBL21677421 0.75 KDM4E (0.42) MAPTLMNAKDM4ECYP1A2CYP3A4
SCHEMBL20740893 0.75 KDM4E (0.42) MAPTLMNAKDM4ECYP1A2CYP3A4
SCHEMBL2649168 0.74 LMNA (0.58) MAPTLMNAKDM4ECYP1A2CYP3A4
SCHEMBL13907344 0.73 MAPT (0.73) MAPTLMNAKDM4ECYP1A2CYP3A4
SCHEMBL4159679 0.72 TTR (0.32)
SCHEMBL9728 0.71 MAPT (1.00) MAPTLMNAKDM4ECYP1A2CYP3A4
SCHEMBL7713106 0.71 LMNA (0.48) MAPTLMNACYP1A2CYP3A4NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009068885-A1 DINUCLEAR, QUADRUPLY-STRANDED COMPOUNDS COMPRISING PALLADIUM OR PLATINUM THE UNIVERSITY OF BIRMINGHAM (GB) 2009-06-04 WO disclosed