SCHEMBL4380177

SCHEMBL4380177

Cn1c(SCCCN2CCc3cc(C(F)(F)F)ccc3C2)nnc1-c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 20/20 0.64
DRD2 P14416 15/20 0.64
KCNH2 Q12809 12/20 0.64
HRH1 P35367 2/20 0.61
HTR1A P08908 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7204494 0.99 DRD3 (0.63) DRD3DRD2KCNH2HRH1
SCHEMBL4382046 0.96 DRD3 (0.64) DRD3DRD2KCNH2HRH1HTR1A
Hydrochloric Acid SCHEMBL7203533 0.95 DRD3 (0.63) DRD3DRD2KCNH2HRH1
SCHEMBL4387226 0.88 DRD3 (0.61) DRD3DRD2KCNH2HRH1
Hydrochloric Acid SCHEMBL7205784 0.87 DRD3 (0.60) DRD3DRD2KCNH2HRH1
SCHEMBL4389064 0.86 DRD3 (0.69) DRD3DRD2KCNH2HRH1HTR1A
SCHEMBL4390849 0.86 DRD3 (0.62) DRD3DRD2KCNH2HRH1HTR1A
Hydrochloric Acid SCHEMBL7201490 0.85 DRD3 (0.61) DRD3DRD2KCNH2HRH1HTR1A
SCHEMBL4387221 0.84 DRD3 (0.62) DRD3DRD2KCNH2HRH1HTR1A
SCHEMBL4386717 0.84 DRD3 (0.61) DRD3DRD2KCNH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed