SCHEMBL4384802

SCHEMBL4384802

Cn1c(SCCCN2CCc3ccc(S(=O)(=O)Nc4ccccc4)cc3C2)nnc1-c1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 19/20 0.54
KCNH2 Q12809 8/20 0.54
DRD2 P14416 17/20 0.49
CYP3A4 P08684 1/20 0.47
CHRM1 P11229 1/20 0.47
CHRM3 P20309 1/20 0.47
ALDH1A1 P00352 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4388088 0.93 DRD3 (0.55) DRD3KCNH2DRD2ALDH1A1
SCHEMBL4395457 0.90 DRD3 (0.52) DRD3KCNH2DRD2CYP3A4CHRM1
SCHEMBL4386866 0.85 DRD3 (0.55) DRD3KCNH2DRD2CYP3A4CHRM1
SCHEMBL4385575 0.83 DRD3 (0.45) DRD3KCNH2DRD2
Hydrochloric Acid SCHEMBL7202732 0.82 DRD3 (0.64) DRD3KCNH2DRD2CYP3A4CHRM1
SCHEMBL4562741 0.82 DRD3 (0.53) DRD3KCNH2DRD2CYP3A4CHRM1
SCHEMBL4387200 0.82 DRD3 (0.58) DRD3KCNH2DRD2ALDH1A1
SCHEMBL4702317 0.82 DRD3 (0.56) DRD3KCNH2DRD2CYP3A4CHRM1
SCHEMBL4381620 0.81 DRD3 (0.50) DRD3KCNH2DRD2CYP3A4CHRM1
SCHEMBL4392618 0.81 DRD3 (0.57) DRD3KCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed
US-6602867-B1 Triazole compounds with dopamine-D3-receptor affinity ABBOTT LABORATORIES 2003-08-05 US disclosed