SCHEMBL4386446

SCHEMBL4386446

COc1cccc(-c2cccc(C3(c4ccncc4)N=C(N)c4cccnc43)c2F)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.47
BACE2 Q9Y5Z0 7/20 0.44
CTSD P07339 6/20 0.44
KCNH2 Q12809 6/20 0.43
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3776518 0.82 BACE1 (0.59) BACE1BACE2CTSDKCNH2
SCHEMBL4386451 0.77 KDM1A (0.39) BACE1BACE2CTSDKCNH2PDE4A
SCHEMBL3548391 0.77 BACE1 (0.71) BACE1BACE2CTSDKCNH2
SCHEMBL3847650 0.75 BACE1 (0.63) BACE1BACE2CTSDKCNH2
SCHEMBL3636805 0.74 BACE1 (0.57) BACE1BACE2CTSDKCNH2
SCHEMBL2087395 0.74 BACE1 (0.60) BACE1BACE2CTSDKCNH2
SCHEMBL3633227 0.74 BACE1 (0.58) BACE1BACE2CTSDKCNH2
SCHEMBL2084648 0.73 BACE1 (0.62) BACE1BACE2CTSDKCNH2
Trifluoroacetic Acid SCHEMBL2085922 0.73 BACE1 (0.59) BACE1BACE2CTSDKCNH2
SCHEMBL3243720 0.72 BACE1 (0.48) BACE1BACE2CTSDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629356-B2 Substituted pyrrolo[3,4-b]pyridinamines and pharmaceutical compositions ASTRAZENECA AB (SE) 2009-12-08 US disclosed