SCHEMBL4386451

SCHEMBL4386451

COc1cccc(-c2cccc(C3(c4ccncc4)NC(N)c4cccnc43)c2F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.39
KDM1B Q8NB78 2/20 0.39
BACE1 P56817 5/20 0.39
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
KCNH2 Q12809 1/20 0.38
KDR P35968 1/20 0.37
RPS6KA3 P51812 1/20 0.36
CTSD P07339 3/20 0.36
DYRK1A Q13627 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
BACE2 Q9Y5Z0 2/20 0.35
GCGR P47871 1/20 0.35
MAPK14 Q16539 1/20 0.35
NTRK1 P04629 1/20 0.35
MGAT2 Q10469 1/20 0.34
DHODH Q02127 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3776523 0.84 BACE1 (0.46) KDM1ABACE1CTSDBACE2DHODH
SCHEMBL3847657 0.78 BACE1 (0.47) BACE1CTSDBACE2MAPT
SCHEMBL4386446 0.77 BACE1 (0.47) BACE1PDE4APDE4BPDE4CPDE4D
SCHEMBL3636810 0.74 BACE1 (0.46) KDM1ABACE1KCNH2CTSDBACE2
SCHEMBL3633229 0.74 BACE1 (0.46) KDM1AKDM1BBACE1PDE4APDE4B
SCHEMBL3243724 0.72 KDM1A (0.40) KDM1ABACE1PDE4APDE4BPDE4C
SCHEMBL4398010 0.71 TEK (0.36) BACE1KCNH2RPS6KA3CTSDBACE2
SCHEMBL3785651 0.70 BACE1 (0.42) BACE1KCNH2BACE2
SCHEMBL3773671 0.69 CHRNA1 (0.32)
SCHEMBL3780604 0.69 BACE1 (0.46) BACE1CTSDBACE2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629356-B2 Substituted pyrrolo[3,4-b]pyridinamines and pharmaceutical compositions ASTRAZENECA AB (SE) 2009-12-08 US disclosed