SCHEMBL43865

SCHEMBL43865

Cc1ccccc1C[C@H](N)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.59
NOS1 P29475 3/20 0.59
NOS2 P35228 3/20 0.59
SLC7A5 Q01650 3/20 0.58
PKM P14618 2/20 0.58
ALPI P09923 1/20 0.58
PTGS1 P23219 1/20 0.58
XIAP P98170 1/20 0.58
MAPT P10636 3/20 0.51
KDM4E B2RXH2 2/20 0.51
MEN1 O00255 2/20 0.51
LMNA P02545 2/20 0.51
BLM P54132 2/20 0.51
PMP22 Q01453 2/20 0.51
KMT2A Q03164 2/20 0.51
HIF1A Q16665 2/20 0.51
MPO P05164 1/20 0.51
TSHR P16473 1/20 0.51
ALDH1A1 P00352 2/20 0.50
RECQL P46063 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL43864 1.00 NOS3 (0.59) NOS3NOS1NOS2SLC7A5PKM
SCHEMBL383453 1.00 NOS3 (0.59) NOS3NOS1NOS2SLC7A5PKM
SCHEMBL29379111 1.00 NOS3 (0.59) NOS3NOS1NOS2SLC7A5PKM
Hydrochloric Acid SCHEMBL28690926 0.98 NOS3 (0.58) NOS3NOS1NOS2SLC7A5PKM
Hydrochloric Acid SCHEMBL28690928 0.98 NOS3 (0.58) NOS3NOS1NOS2SLC7A5PKM
Dl-Phenylalanine SCHEMBL23214377 0.93 SLC7A5 (0.71) NOS3NOS1NOS2SLC7A5PKM
SCHEMBL27464327 0.87 NOS3 (0.48) NOS3NOS1NOS2SLC7A5PKM
SCHEMBL13971424 0.86 SLC7A5 (0.69) NOS3NOS1NOS2SLC7A5PKM
SCHEMBL9164980 0.86 SLC7A5 (0.69) NOS3NOS1NOS2SLC7A5PKM
SCHEMBL5326602 0.86 NOS3 (0.53) NOS3NOS1NOS2SLC7A5PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2369 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250325672-A1 ANTI-INFECTIVE BICYCLIC PEPTIDE LIGANDS BICYCLE TX LTD (GB) 2025-10-23 US claimed
EP-4619043-A1 FIBROBLAST ACTIVATION PROTEIN TARGETED COMPOUNDS AND USE THEREOF Perspective Therapeutics, Inc. (US) 2025-09-24 EP claimed
WO-2025128149-A1 FIBROBLAST ACTIVATION PROTEIN TARGETED COMPOUNDS AND USE THEREOF VIEWPOINT MOLECULAR TARGETING, INC. (US) 2025-06-19 WO claimed
US-20250186630-A1 FIBROBLAST ACTIVATION PROTEIN TARGETING PEPTIDES VIEWPOINT MOLECULAR TARGETING, INC. (US) 2025-06-12 US claimed
WO-2025094171-A1 SUPERHYDROPHOBIC COATING YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2025-05-08 WO claimed
CN-118406439-B Chemical mechanical polishing composition and application thereof in tungsten chemical mechanical polishing 万华化学集团电子材料有限公司 2024-10-18 CN claimed
CN-114457049-B Pyrrolysiyl-tRNA synthetase mutant and application thereof 浙江大学杭州国际科创中心 2024-09-24 CN claimed
CN-118406439-A Chemical mechanical polishing composition and application thereof in tungsten chemical mechanical polishing 万华化学集团电子材料有限公司 2024-07-30 CN claimed
US-11904020-B2 Bicyclic peptide ligands specific for TREM2 BICYCLETX LIMITED (GB) 2024-02-20 US claimed
EP-4308586-A1 BICYCLIC PEPTIDE LIGANDS SPECIFIC FOR TREM2 BicycleTX Limited (GB) 2024-01-24 EP claimed
WO-2003037916-A2 LINEAR BASIC COMPOUNDS HAVING NK-2 ANTAGONIST ACTIVITY AND FORMULATIONS THEREOF MALESCI ISTITUTO FARMACOBIOLOGICO S.P.A. (IT) 2003-05-08 WO claimed
EP-0918534-A4 PEPTIDYL PRODRUGS AND METHODS OF MAKING AND USING THE SAME UNIV PITTSBURGH (US) 2001-10-10 EP claimed
EP-1046627-A2 Enantiopure reagents and process for the separation of enantiomers SOLVAY (Société Anonyme) (BE) 2000-10-25 EP claimed
US-5952294-A OLIGOPEPTIDE ATTACHED TO AMINO, HYDROXY OR THIOL FUNCTIONS OF THERAPEUTIC AGENT, E.G. ARA-C, TO EXTEND ITS BIOLOGICAL ACTIVE LIVE IN VIVO; CONTROLLING THE KINETICS AND METABOLISM; LEUKEMIA; VIRICIDES; ANTITUMOR/-CARCINOGENIC AGENTS UNIVERSITY OF PITTSBURGH OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 1999-09-14 US claimed
EP-0920307-A2 DERIVATES FROM BISARYLTETRACARBONACID, AND PHARMARCEUTICAL PRODUCT CONTAINING THEM Roche Diagnostics GmbH (DE) 1999-06-09 EP claimed
EP-0918534-A1 PEPTIDYL PRODRUGS AND METHODS OF MAKING AND USING THE SAME UNIVERSITY OF PITTSBURGH OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 1999-06-02 EP claimed
WO-1998006386-A2 DERIVATES FROM BISARYLTETRACARBONACID, AND PHARMARCEUTICAL PRODUCT CONTAINING THEM ROCHE DIAGNOSTICS GMBH (DE) 1998-02-19 WO claimed
WO-1998004277-A1 PEPTIDYL PRODRUGS AND METHODS OF MAKING AND USING THE SAME UNIVERSITY OF PITTSBURGH OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 1998-02-05 WO claimed
EP-0352092-B1 Novel antibiotics R106 TAKARA SHUZO CO (JP) 1993-10-27 EP claimed
EP-0352092-A2 Novel antibiotics R106 TAKARA SHUZO CO. LTD. (JP) 1990-01-24 EP claimed