SCHEMBL4386594

SCHEMBL4386594

COc1ccc2c(c1)c(C(=O)C(=O)Nc1ccnc(Cl)c1)c(C)n2Cc1ccc(Cl)cc1.COc1ccc2c(c1)c(C(=O)C(=O)Nc1ccnc(Cl)c1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.70
PLA2G2A P14555 6/20 0.50
MAPT P10636 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ALDH1A1 P00352 2/20 0.50
RGS12 O14924 1/20 0.50
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
PKM P14618 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
MAPK1 P28482 1/20 0.50
CYP2C19 P33261 1/20 0.50
GNAI1 P63096 1/20 0.50
PMP22 Q01453 1/20 0.50
HIF1A Q16665 1/20 0.50
PTGS2 P35354 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2168496 0.97 FAAH (0.74) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL2168479 0.96 FAAH (0.62) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL2160463 0.93 FAAH (0.68) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL2159703 0.90 FAAH (0.64) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL3005475 0.90 FAAH (0.64) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL2159916 0.89 FAAH (0.87) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL2159931 0.89 FAAH (0.68) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL9952751 0.89 FAAH (0.73) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL2167924 0.89 FAAH (0.54) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL2168973 0.88 FAAH (0.72) FAAHPLA2G2AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed