SCHEMBL4386795

SCHEMBL4386795

COc1ccc2c(c1F)c(CC(=O)OC(=O)C(C)c1c(C)n(C(=O)c3ccc(Cl)cc3)c3ccc(O)c(F)c13)c(C)n2C(=O)c1ccc(Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.45
CNR2 P34972 1/20 0.43
AKR1C3 P42330 1/20 0.43
PTGS1 P23219 2/20 0.42
HTR1A P08908 1/20 0.42
PKM P14618 1/20 0.42
GLO1 Q04760 1/20 0.42
HIF1A Q16665 1/20 0.42
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4386800 0.88 PTGS2 (0.50) PTGS2AKR1C3PTGS1HTR1APKM
SCHEMBL12255241 0.82 PTGS2 (0.62) PTGS2CNR2AKR1C3PTGS1HTR1A
SCHEMBL5797673 0.81 PTGS2 (0.43) PTGS2AKR1C3PTGS1
SCHEMBL5797670 0.81 PTGS2 (0.43) PTGS2AKR1C3PTGS1
SCHEMBL2004898 0.80 PTGS2 (0.46) PTGS2AKR1C3PTGS1GLO1HIF1A
SCHEMBL5797099 0.80 PTGS2 (0.40) PTGS2AKR1C3PTGS1
SCHEMBL5798162 0.79 AKR1C3 (0.47) PTGS2AKR1C3PTGS1HTR1APKM
SCHEMBL5799946 0.79 PTGS2 (0.43) PTGS2AKR1C3PTGS1GLO1HIF1A
SCHEMBL5799952 0.79 PTGS2 (0.43) PTGS2AKR1C3PTGS1GLO1HIF1A
SCHEMBL3004878 0.79 PTGS2 (0.63) PTGS2AKR1C3PTGS1HTR1APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2610244-A1 Indole compounds Ironwood Pharmaceuticals, Inc. (US) 2013-07-03 EP disclosed
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed