SCHEMBL4388576

SCHEMBL4388576

CC(C)(C)OC(=O)N1C[C@H](NCc2ccccc2)C[C@H]1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 4/20 0.48
HDAC8 Q9BY41 1/20 0.42
HTRA1 Q92743 1/20 0.42
KMT2A Q03164 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ACE P12821 3/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
STS P08842 1/20 0.40
MCL1 Q07820 1/20 0.40
ACHE P22303 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
NAMPT P43490 1/20 0.40
BCHE P06276 1/20 0.40
BACE1 P56817 1/20 0.40
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29548635 0.93 ACE (0.45) AGTR2HTRA1KMT2AACEMCL1
SCHEMBL13841901 0.91 MMP2 (0.47) AGTR2HDAC8HTRA1KMT2AL3MBTL1
SCHEMBL24538202 0.91 MMP2 (0.47) AGTR2HDAC8HTRA1KMT2AL3MBTL1
SCHEMBL12166250 0.91 MMP2 (0.47) AGTR2HDAC8HTRA1KMT2AL3MBTL1
SCHEMBL2824741 0.91 MMP2 (0.47) AGTR2HDAC8HTRA1KMT2AL3MBTL1
SCHEMBL13548957 0.88 CARM1 (0.47) AGTR2HDAC8NR1H2NR1H3
SCHEMBL8254788 0.88 CARM1 (0.47) AGTR2HDAC8NR1H2NR1H3
SCHEMBL29548707 0.88 NR1H2 (0.42) AGTR2NAMPTNR1H2
SCHEMBL8936138 0.87 KMT2A (0.42) HDAC8KMT2AL3MBTL1JAK2JAK1
SCHEMBL29548674 0.86 USP30 (0.45) AGTR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1950199-B1 Proline derivatives and use thereof as drugs MITSUBISHI TANABE PHARMA CORP (JP) 2009-12-02 EP disclosed