SCHEMBL4388807

SCHEMBL4388807

CC(C)c1cc(-c2ncoc2-c2ccc(NCCN3CCOCC3)cc2)c(O)cc1O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 14/20 0.47
HSP90AB1 P08238 7/20 0.47
PDK1 Q15118 1/20 0.44
TRAP1 Q12931 3/20 0.44
HSP90B1 P14625 2/20 0.44
EGFR P00533 1/20 0.42
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4245797 0.84 MEN1 (0.50) HSP90AA1HSP90AB1PDK1TRAP1HSP90B1
SCHEMBL4063737 0.84 PDK1 (0.58) HSP90AA1HSP90AB1PDK1TRAP1HSP90B1
SCHEMBL13847844 0.82 TLR9 (0.42) EGFRKDM4ETLR9TLR8TLR7
SCHEMBL4069471 0.81 EGFR (0.43) EGFRKDM4ERAB9ATLR9TLR8
SCHEMBL4238978 0.80 PDK1 (0.43) HSP90AA1HSP90AB1PDK1TRAP1HSP90B1
SCHEMBL4385992 0.76 HSP90AA1 (0.56) HSP90AA1HSP90AB1PDK1TRAP1HSP90B1
SCHEMBL4395463 0.76 HSP90AA1 (0.54) HSP90AA1HSP90AB1PDK1TRAP1HSP90B1
SCHEMBL4062363 0.76 MAPK14 (0.48) HSP90AA1HSP90AB1
SCHEMBL28934605 0.75 HSP90AA1 (0.45) HSP90AA1HSP90AB1
SCHEMBL4397076 0.75 HSP90AA1 (0.55) HSP90AA1HSP90AB1PDK1TRAP1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009066060-A2 4-SUBSTITUTED-6-ISOPROPYL-BENZENE-1,3-DIOL COMPOUNDS AND THEIR USE TOPOTARGET A/S (DK) 2009-05-28 WO disclosed
WO-2009066060-A2 4-SUBSTITUTED-6-ISOPROPYL-BENZENE-1,3-DIOL COMPOUNDS AND THEIR USE TOPOTARGET A/S (DK) 2009-05-28 WO disclosed