SCHEMBL4392886

SCHEMBL4392886

CC(C)(C)OC(=O)N1C[C@@H](Nc2ncccc2C(F)(F)F)C[C@H]1C(=O)N1CCSC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
HSD11B1 P28845 2/20 0.41
CYP2D6 P10635 1/20 0.41
TRPV1 Q8NER1 2/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
PREP P48147 1/20 0.36
GAA P10253 1/20 0.36
WNT3 P56703 2/20 0.36
SFRP1 Q8N474 2/20 0.36
DPP4 P27487 2/20 0.35
TGM2 P21980 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
SSTR4 P31391 4/20 0.35
SSTR1 P30872 2/20 0.35
POLB P06746 1/20 0.35
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35
ERBB3 P21860 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2708987 0.82 DPP4 (0.42) CYP3A4CYP2C9HSD11B1CYP2D6TRPV1
SCHEMBL2709311 0.81 DPP4 (0.53) PREPDPP4TGM2
SCHEMBL2709313 0.81 DPP4 (0.53) PREPDPP4TGM2
SCHEMBL2709711 0.80 DPP4 (0.51) CYP3A4CYP2C9HSD11B1CYP2D6TRPV1
SCHEMBL2709717 0.80 DPP4 (0.51) CYP3A4CYP2C9HSD11B1CYP2D6TRPV1
SCHEMBL2708647 0.79 DPP4 (0.40) PREPWNT3SFRP1DPP4TGM2
SCHEMBL4392882 0.79 PREP (0.39) CYP3A4PREPDPP4TGM2POLB
SCHEMBL2709456 0.78 DPP4 (0.55) PREPDPP4
SCHEMBL2709078 0.77 DPP4 (0.59) PREPDPP4
SCHEMBL2709196 0.77 DPP4 (0.58) CYP3A4CYP2C9HSD11B1CYP2D6DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1950199-B1 Proline derivatives and use thereof as drugs MITSUBISHI TANABE PHARMA CORP (JP) 2009-12-02 EP disclosed