SCHEMBL4393480

SCHEMBL4393480

Cn1c(CN2CCNCC2=O)cc2cnccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 5/20 0.49
CDK4 P11802 1/20 0.39
CDK6 Q00534 1/20 0.39
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
MKNK2 Q9HBH9 4/20 0.35
KDM4E B2RXH2 1/20 0.33
PRKD3 O94806 1/20 0.33
PRKCG P05129 1/20 0.33
CYP1A2 P05177 1/20 0.33
PRKCB P05771 1/20 0.33
CYP3A4 P08684 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
PRKCA P17252 1/20 0.33
PRKACA P17612 1/20 0.33
PRKACG P22612 1/20 0.33
PRKACB P22694 1/20 0.33
PRKCH P24723 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27591557 0.84 F10 (0.43) F10CDK4CDK6JAK2JAK1
SCHEMBL27526854 0.83 F10 (0.38) F10CDK4CDK6JAK2JAK1
SCHEMBL1652849 0.80 F10 (0.36) F10CDK4CDK6
SCHEMBL27572912 0.80 F10 (0.36) F10CDK4CDK6JAK2JAK1
SCHEMBL4397329 0.74 F10 (0.51) F10CDK4CDK6
SCHEMBL14993193 0.71 ALDH1A1 (0.53) CDK4CDK6KDM4E
Hydrochloric Acid SCHEMBL1306753 0.70 ALDH1A1 (0.52) CDK4CDK6KDM4E
SCHEMBL23460609 0.69 MAPK1 (0.48) F10KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL23461159 0.68 CYP2A6 (0.40) F10KDM4E
Tert-Butyl Formate SCHEMBL27572914 0.68 F10 (0.45) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612075-B2 Substituted oxoazaheterocyclyl compounds AVENTIS PHARMACEUTICALS INC. (US) 2009-11-03 US disclosed
US-7612075-B2 Substituted oxoazaheterocyclyl compounds AVENTIS PHARMACEUTICALS INC. (US) 2009-11-03 US disclosed
US-7612075-B2 Substituted oxoazaheterocyclyl compounds AVENTIS PHARMACEUTICALS INC. (US) 2009-11-03 US disclosed