SCHEMBL4394150

SCHEMBL4394150

NC(=NO)c1ccc2c(c1)CNC(=O)N2

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.49
PDE3A Q14432 2/20 0.49
CYP11B1 P15538 2/20 0.44
CYP11B2 P19099 2/20 0.44
CRBN Q96SW2 2/20 0.38
MAPK1 P28482 1/20 0.36
RECQL P46063 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
KCNH2 Q12809 1/20 0.34
MB P02144 1/20 0.34
SMYD3 Q9H7B4 3/20 0.32
KDM1A O60341 3/20 0.32
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4405787 0.88 PDE3B (0.39) PDE3BPDE3ACYP11B1CYP11B2CRBN
SCHEMBL4399635 0.82 PDE3B (0.51) PDE3BPDE3ACYP11B1CYP11B2CRBN
SCHEMBL1519694 0.79 SMYD3 (0.50) PDE3BPDE3ASMYD3
SCHEMBL1519697 0.79 SMYD3 (0.50) PDE3BPDE3ASMYD3
SCHEMBL5366326 0.78 PDE3B (0.54) PDE3BPDE3ACYP11B1CYP11B2CRBN
SCHEMBL31032797 0.78 PDE3B (0.54) PDE3BPDE3ACYP11B1CYP11B2CRBN
SCHEMBL4397716 0.75 CYP11B1 (0.44) PDE3BPDE3ACYP11B1CYP11B2RECQL
SCHEMBL4394147 0.73 PDE3B (0.49) PDE3BPDE3ACYP11B1CYP11B2CRBN
SCHEMBL18114133 0.73 PDE3B (0.49) PDE3BPDE3ACYP11B1CYP11B2CRBN
SCHEMBL16548893 0.73 PDE3B (0.60) PDE3BPDE3ACYP11B1CYP11B2CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed