SCHEMBL4397716

SCHEMBL4397716

NC(=NO)c1ccc2c(c1)COC(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.44
CYP11B2 P19099 2/20 0.44
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
SYK P43405 1/20 0.36
KCNH2 Q12809 1/20 0.35
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
RECQL P46063 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
CTSC P53634 1/20 0.33
CPT2 P23786 2/20 0.32
CPT1A P50416 2/20 0.32
CPT1B Q92523 1/20 0.32
SMYD3 Q9H7B4 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4395266 0.82 CYP11B1 (0.46) CYP11B1CYP11B2PDE3BPDE3ASYK
SCHEMBL25184590 0.78 CYP11B1 (0.47) CYP11B1CYP11B2PDE3BPDE3ASYK
SCHEMBL1519697 0.78 SMYD3 (0.50) PDE3BPDE3ASMYD3GRIA1HDAC3
SCHEMBL1519694 0.78 SMYD3 (0.50) PDE3BPDE3ASMYD3GRIA1HDAC3
SCHEMBL4394150 0.75 PDE3B (0.49) CYP11B1CYP11B2PDE3BPDE3AKCNH2
SCHEMBL1341398 0.75 MAPT (0.54) KCNH2RECQLLMNA
SCHEMBL1341399 0.75 MAPT (0.54) KCNH2RECQLLMNA
SCHEMBL4397712 0.74 CYP11B1 (0.44) CYP11B1CYP11B2PDE3BPDE3ASYK
SCHEMBL10916724 0.73 CYP11B1 (0.51) CYP11B1CYP11B2PDE3BPDE3ASYK
SCHEMBL3597266 0.73 LMNA (0.51) CYP11B1CYP11B2PDE3BPDE3ASYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed