SCHEMBL439457

SCHEMBL439457

CCOC(=O)c1cnc2c(C)cc(C)cc2c1N

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
KMT2A Q03164 2/20 0.57
THRB P10828 2/20 0.56
MAPT P10636 3/20 0.52
GAA P10253 1/20 0.51
RAD52 P43351 1/20 0.51
UHRF1 Q96T88 1/20 0.51
HSP90AA1 P07900 1/20 0.48
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
TP53 P04637 1/20 0.45
DPP4 P27487 2/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL438293 0.87 NPC1 (0.55) NPC1RAB9AKMT2ATHRBMAPT
SCHEMBL437001 0.87 NPC1 (0.55) NPC1RAB9AKMT2ATHRBGAA
SCHEMBL441793 0.87 TP53 (0.56) NPC1RAB9AKMT2ATHRBMAPT
SCHEMBL438821 0.87 KMT2A (0.55) NPC1RAB9AKMT2ATHRBMAPT
SCHEMBL11240555 0.85 THRB (0.57) NPC1RAB9AKMT2ATHRBMAPT
SCHEMBL17524914 0.84 THRB (0.56) NPC1RAB9AKMT2ATHRBMAPT
SCHEMBL11242678 0.84 KMT2A (0.57) NPC1RAB9AKMT2ATHRBMAPT
SCHEMBL437086 0.81 KDM4E (0.53) KMT2ATHRBMAPTGAARAD52
SCHEMBL438878 0.81 KMT2A (0.71) NPC1RAB9AKMT2AMAPTGAA
SCHEMBL438415 0.79 KMT2A (0.55) NPC1RAB9AKMT2AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed