SCHEMBL4394807

SCHEMBL4394807

Cn1c(C(=O)NCCCCN2CCc3ccc(S(=O)(=O)N4CCCC4)cc3C2)nnc1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.49
DRD3 P35462 10/20 0.49
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 1/20 0.46
DRD1 P21728 1/20 0.45
DRD4 P21917 1/20 0.45
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
RECQL P46063 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 1/20 0.44
HTT P42858 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
ACKR3 P25106 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4382332 0.86 KDM4E (0.46) DRD2DRD3KDM4EALDH1A1HPGD
SCHEMBL4381610 0.82 KDM4E (0.44) DRD2DRD3KDM4EALDH1A1HPGD
SCHEMBL4392626 0.81 DRD3 (0.58) DRD2DRD3KDM4EALDH1A1HPGD
SCHEMBL4394660 0.81 DRD3 (0.60) DRD2DRD3KDM4EALDH1A1HPGD
SCHEMBL4385475 0.81 DRD3 (0.60) DRD2DRD3KDM4EALDH1A1HPGD
SCHEMBL4386303 0.77 DRD3 (0.55) DRD2DRD3KDM4EALDH1A1HPGD
SCHEMBL4392739 0.76 HTT (0.42) DRD2DRD3KDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL7199896 0.75 HTT (0.41) DRD2DRD3KDM4EALDH1A1HPGD
SCHEMBL4380366 0.75 DRD3 (0.54) DRD2DRD3KDM4EALDH1A1HPGD
SCHEMBL4380463 0.75 DRD3 (0.55) DRD2DRD3KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed
US-6602867-B1 Triazole compounds with dopamine-D3-receptor affinity ABBOTT LABORATORIES 2003-08-05 US disclosed