SCHEMBL4381610

SCHEMBL4381610

Cn1c(CCCCN2CCc3ccc(S(=O)(=O)N4CCCCC4)cc3C2)nnc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.44
ALDH1A1 P00352 6/20 0.44
HPGD P15428 3/20 0.44
HRH3 Q9Y5N1 2/20 0.44
HSD17B10 Q99714 2/20 0.41
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MAPT P10636 1/20 0.40
GBA1 P04062 2/20 0.39
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39
GAA P10253 2/20 0.39
TSHR P16473 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
KCNH2 Q12809 1/20 0.39
HTT P42858 1/20 0.39
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4392739 0.92 HTT (0.42) KDM4EALDH1A1HPGDHSD17B10HTR2C
Hydrochloric Acid SCHEMBL7199896 0.91 HTT (0.41) KDM4EALDH1A1HPGDHSD17B10HTR2C
SCHEMBL4395639 0.89 HTR7 (0.43) DRD2DRD3KCNH2HTR7
SCHEMBL4385475 0.85 DRD3 (0.60) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL4394660 0.85 DRD3 (0.60) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL4382332 0.84 KDM4E (0.46) KDM4EALDH1A1HPGDHRH3HSD17B10
SCHEMBL4392626 0.84 DRD3 (0.58) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL4394807 0.82 DRD2 (0.49) KDM4EALDH1A1HPGDDRD2DRD3
SCHEMBL4386303 0.79 DRD3 (0.55) KDM4EALDH1A1HPGDHSD17B10HTR2C
SCHEMBL4543121 0.78 DRD2 (0.57) HTR2BDRD2DRD3KCNH2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed
US-6602867-B1 Triazole compounds with dopamine-D3-receptor affinity ABBOTT LABORATORIES 2003-08-05 US disclosed