SCHEMBL4395877

SCHEMBL4395877

NCc1cccc(C2CCN(C(=O)c3cc4ccccc4s3)CC2)c1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 6/20 0.55
HRH4 Q9H3N8 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
CAPN1 P07384 1/20 0.52
CTSB P07858 1/20 0.52
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
KCNH2 Q12809 1/20 0.51
CCR1 P32246 1/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1386521 0.93 TPSAB1 (0.60) TPSAB1
SCHEMBL15772184 0.85 CYP3A4 (0.53) TPSAB1CYP3A4CYP2D6KCNH2
SCHEMBL15780781 0.84 TPSAB1 (0.54) TPSAB1CYP3A4CYP2D6KCNH2
Trifluoroacetic Acid SCHEMBL4409332 0.82 TPSAB1 (0.55) TPSAB1
Trifluoroacetic Acid SCHEMBL4412717 0.82 TPSAB1 (0.55) TPSAB1
SCHEMBL18652739 0.81 TPSAB1 (0.52) TPSAB1CYP3A4CYP2D6KCNH2
SCHEMBL15788544 0.81 TPSAB1 (0.52) TPSAB1CYP3A4CYP2D6KCNH2
SCHEMBL15788466 0.80 TPSAB1 (0.50) TPSAB1CYP3A4CYP2D6KCNH2
Trifluoroacetic Acid SCHEMBL4395571 0.79 TPSAB1 (0.59) TPSAB1
SCHEMBL1384467 0.79 TPSAB1 (0.53) TPSAB1CYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-B1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMA INC (US) 2009-12-23 EP claimed