SCHEMBL4396897

SCHEMBL4396897

CC(C)NCCNc1ccc(S(=O)(=O)Oc2ccc3nc(NC(=O)CCC4CCNCC4)sc3c2)cc1.O=C(CCC1CCNCC1)Nc1nc2ccc(OS(=O)(=O)c3ccc(NCCCn4ccnc4)cc3)cc2s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 4/20 0.46
NPC1 O15118 3/20 0.39
ALDH1A1 P00352 2/20 0.37
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TSHR P16473 1/20 0.36
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPT P10636 1/20 0.35
CASP2 P42575 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4394552 0.95 QPCT (0.49) QPCTNPC1ALDH1A1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL4394550 0.94 QPCT (0.48) QPCTNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL4396985 0.91 ALDH1A1 (0.43) NPC1ALDH1A1RAB9ASMN1; SMN2TSHR
Hydrochloric Acid SCHEMBL4396982 0.90 ALDH1A1 (0.43) NPC1ALDH1A1RAB9ASMN1; SMN2TSHR
SCHEMBL4396959 0.88 QPCT (0.50) QPCTNPC1ALDH1A1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL4396954 0.88 QPCT (0.49) QPCTNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL4394584 0.84 ALDH1A1 (0.52) NPC1ALDH1A1RAB9ASMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL4394580 0.84 ALDH1A1 (0.51) NPC1ALDH1A1RAB9ASMN1; SMN2LMNA
SCHEMBL4399661 0.82 ALDH1A1 (0.44) NPC1ALDH1A1RAB9ASMN1; SMN2TSHR
SCHEMBL4397343 0.82 ALDH1A1 (0.43) NPC1ALDH1A1RAB9ASMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632952-B2 4-(2-hydroxy-2-methylpropylamino)benzenesulfonic acid 2-[(piperidine-4-carbonyl)-amino]benzothiazol-6-yl ester; anticancer activity, via modulation of the activity of proteins, in particular of kinases; anticarcinogenic agent AVENTIS PHARMA S.A. (FR) 2009-12-15 US claimed