SCHEMBL4397987

SCHEMBL4397987

C[C@@H](Oc1cc(-n2cnc3cc(Br)c(OC4CCN(C(=O)O)C(C(C)(C)CF)C4)cc32)sc1C(N)=O)c1ccccc1Cl

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 16/20 0.58
PLK3 Q9H4B4 14/20 0.58
NEK2 P51955 3/20 0.58
PIK3CD O00329 2/20 0.58
NUAK1 O60285 2/20 0.58
PDGFRB P09619 2/20 0.58
PIM1 P11309 2/20 0.58
KDR P35968 2/20 0.58
CDK2 P24941 1/20 0.57
IKBKE Q14164 1/20 0.57
CYP2C9 P11712 3/20 0.51
CYP3A4 P08684 3/20 0.51
PIK3CG P48736 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5003095 0.85 PLK1 (0.62) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4398312 0.83 PLK1 (0.65) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4400487 0.77 PLK1 (0.66) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4397911 0.76 PLK1 (0.56) PLK1PLK3NEK2PIK3CDNUAK1
Gsk-237701A SCHEMBL4034890 0.74 PLK1 (1.00) PLK1PLK3NEK2PIK3CDNUAK1
Gsk-237701A SCHEMBL29644977 0.74 PLK1 (1.00) PLK1PLK3NEK2PIK3CDNUAK1
Gsk-237701A SCHEMBL5065885 0.74 PLK1 (1.00) PLK1PLK3NEK2PIK3CDNUAK1
Gsk-579289A SCHEMBL31060734 0.74 PLK1 (1.00) PLK1PLK3NEK2PIK3CDNUAK1
Gsk-579289A SCHEMBL13206401 0.74 PLK1 (1.00) PLK1PLK3NEK2PIK3CDNUAK1
Gsk-579289A SCHEMBL2989105 0.74 PLK1 (1.00) PLK1PLK3NEK2PIK3CDNUAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924572-B1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SMITHKLINE BEECHAM CORP (US) 2009-12-30 EP disclosed